Product Name | Cobimetinib (GDC-0973; XL518) |
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CAS | 934660-93-2 |
Formula | C21H21F3IN3O2 |
MW | 531.31 |
Appearance | Off-white solid powder |
Storage condition | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
Size | Availability | Price(USD) | VIP Price (USD) | Quantity |
---|---|---|---|---|
5 mg | In-stock | $450.00 | Visible after login | |
10 mg | In-stock | $510.00 | Visible after login | |
50 mg | In-stock | $1200.00 | Visible after login |
Product Name | Cobimetinib (GDC-0973; XL518) |
---|---|
CAS | 934660-93-2 |
Formula | C21H21F3IN3O2 |
MW | 531.31 |
Appearance | Off-white solid powder |
Storage condition | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
Cobimetinib (GDC-0973, RG7420) is a potent and highly selective MEK1 inhibitor with IC50 of 4.2 nM, and showing no significant inhibition when tested against a panel of more than 100 of serine-threonine and tyrosine kinases. Cobimetinib induces apoptosis. Phase 3.