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CPI-0610

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Catalog No：CL2325 CAS No.：1380087-89-7 MDLNo： Formula：C20H16ClN3O2 MW：365.81

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Size	Availability	Price(USD)	VIP Price (USD)	Quantity
5 mg	In-stock	$850.00	Visible after login	- +
10 mg	In-stock	$1360.00	Visible after login	- +

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Product Overview

Product Name	CPI-0610
CAS	1380087-89-7
Formula	C20H16ClN3O2
MW	365.81
Appearance	White to off-white powder
Storage condition	Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).

Product details

Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.

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CL2325

CPI-0610

1380087-89-7 95%