Home > Category > Signaling Pathways > Membrane Transporter/Ion Channel > P-glycoprotein > Tariquidar | XR9576

Tariquidar | XR9576

ChemLeader 98+%

Catalog No：CL2893 CAS No.：206873-63-4 MDLNo： Formula：C38H38N4O6 MW：646.73

Collect Share

Size	Availability	Price(USD)	VIP Price (USD)	Quantity
There is no price information at the moment, you can send an inquiry,and we will reply to you as soon as possible.

Chemical safety data sheet(MSDS)

Download MSDS

Inquiry Add To Cart

Product Overview
Related documents
Product details
Related literature

Product Overview

Product Name	Tariquidar \| XR9576
CAS	206873-63-4
Formula	C38H38N4O6
MW	646.73
Appearance	Off-white to yellow powder
Storage condition	Store in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.

Product details

Tariquidar (XR9576) is a potent and specific inhibitor of P-glycoprotein (P-gp) with the high affinity (K_d=5.1 nM).

Related literature

Simultaneous Semimechanistic Population Analyses of Levofloxacin in Plasma, Lung, and Prostate To Describe the Influence of Efflux Transporters on Drug Distribution following Intravenous and Intratracheal Administration.

PMID: 26621623 PMCID: PMC4750702 DOI: 10.1128/AAC.02317-15

Read more

Regulation of P-glycoprotein expression in brain capillaries in Huntington's disease and its impact on brain availability of antipsychotic agents risperidone and paliperidone.

PMID: 26661162 PMCID: PMC4976744 DOI: 10.1177/0271678X15606459

Read more

Pharmacokinetics of the P-gp Inhibitor Tariquidar in Rats After Intravenous, Oral, and Intraperitoneal Administration.

Read more

Related

Tariquidar dimesylate | XR9576 dimesylate

625375-84-0 98+%

Tariquidar methanesulfonate, hydrate | XR9576 methanesulfonate, hydrate

625375-83-9 98+%

Tariquidar dihydrochloride | XR9576 dihydrochloride

1992047-62-7 98+%

History

Tariquidar | XR9576

206873-63-4 98+%