Home > Category > Signaling Pathways > Epigenetics > Histone Methyltransferase > BIX-01294 trihydrochloride | BIX01294 triHCl

BIX-01294 trihydrochloride | BIX01294 triHCl

ChemLeader 98+%
Catalog No:CL2754A CAS No.:1392399-03-9 MDLNo: Formula:C28H41Cl3N6O2 MW:600.02
Size Availability Price(USD) VIP Price (USD) Quantity

There is no price information at the moment, you can send an inquiry,and we will reply to you as soon as possible.

Chemical safety data sheet(MSDS)

Download MSDS
  • Product Overview
  • Related documents
  • Product details
  • Related literature
Product Overview
Product Name BIX-01294 trihydrochloride | BIX01294 triHCl
CAS1392399-03-9
FormulaC28H41Cl3N6O2
MW600.02
Storage conditionStore in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
Product details

BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM in a cell-free assay, reduces H3K9me2 of bulk histones, also weakly inhibits GLP (primarily H3K9me3), no significant activity observed at other histone methyltransferases. BIX01294 induces autophagy. BIX01294 also inhibits H3K36 methylation by oncoproteins NSD1, NSD2 and NSD3.


Related literature
Sorry, there is no relevant literature
Service
ChemLeader
021-58180488
Online service time: 9:00-18:00 on weekdays